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A convenient synthesis of N-Boc-protected tert-butyl esters of phenylglycines from benzylamines

✍ Scribed by Naoki Kise; Hiroshi Ozaki; Hiroaki Terui; Kengo Ohya; Nasuo Ueda

Publisher
Elsevier Science
Year
2001
Tongue
French
Weight
61 KB
Volume
42
Category
Article
ISSN
0040-4039

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✦ Synopsis

The N,N-di-Boc-protected benzylamines undergo [1,2] Boc migration on treatment with KDA/t-BuOLi. By this reaction, the corresponding N-Boc-protected t-butyl esters of phenylglycines are obtained in high yields.

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