๐”– Bobbio Scriptorium
โœฆ   LIBER   โœฆ

A convenient synthesis of 1,3,4-thiadiazole and 1,3,4-oxadiazole based peptidomimetics employing diacylhydrazines derived from amino acids

โœ Scribed by G. Nagendra; Ravi S. Lamani; N. Narendra; Vommina V. Sureshbabu


Book ID
104098396
Publisher
Elsevier Science
Year
2010
Tongue
French
Weight
280 KB
Volume
51
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.


๐Ÿ“œ SIMILAR VOLUMES


A facile synthesis of N-Z/Boc-protected
โœ Ravi S. Lamani; G. Nagendra; Vommina V. Sureshbabu ๐Ÿ“‚ Article ๐Ÿ“… 2010 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 713 KB

Synthesis of 1,3,4-oxadiazole containing peptidomimetics is described by a p-TsCl/pyridine-mediated cyclization of the corresponding dipeptidyl thiosemicarbazides, which are readily prepared by coupling N-protected amino acid hydrazides with amino acid-derived isothiocyanato esters. Further, the pro