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A concise synthesis of a highly functionalized C-aryl taxol analog by an intramolecular Heck olefination reaction

✍ Scribed by John J. Masters; David K. Jung; William G. Bornmann; Samuel J. Danishefsky; Susan de Gala

Publisher: Elsevier Science
Year: 1993
Tongue: French
Weight: 235 KB
Volume: 34
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(00)79301-4

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✦ Synopsis

A palladium(O) catalyzed intramolecular Heck olefinatbn used to establish the Cl O-Cl 1 connection in a highly functbnalized taxane analog is described.

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