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4-DAMP analogues reveal heterogeneity of M1 muscarinic receptors

โœ Scribed by R. Micheletti; L. Giudici; M. Turconi; A. Donetti


Book ID
117959386
Publisher
Nature Publishing Group
Year
1990
Tongue
English
Weight
514 KB
Volume
100
Category
Article
ISSN
0007-1188

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Heterogeneity of Guinea-Pig Lung Muscari
โœ E.-B. Haddad; A. Trifilieff; Y. Landry; J.-P. Gies ๐Ÿ“‚ Article ๐Ÿ“… 1993 ๐Ÿ› Elsevier ๐ŸŒ English โš– 453 KB

SUMMARY: Muscarinic receptors present in guinea-pig lung were characterized using the \(M_{3}\) selective radioligand \(\left[{ }^{3} \mathrm{H}\right] 4\)-diphenylacetoxy- \(\mathrm{N}\)-methyl-piperidine methiodide \(\left(\left[{ }^{3} \mathrm{H}\right] 4\right.\)-DAMP). In saturation studies, \(