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4-[18F]fluoromethylbenzylsulfonate ester: a rapid and efficient synthetic method for the N-[18F]fluoromethylbenzylation of amides and amines

✍ Scribed by Yearn Seong Choe; Dong Hyuck Song; Lee Kee-Jung; Sang Eun Kim; Choi Yong; Kyung Han Lee; Kim Byung-Tae; Seung Jun Oh; Dae Yoon Chi

Book ID: 108484451
Publisher: Elsevier Science
Year: 1998
Tongue: English
Weight: 404 KB
Volume: 49
Category: Article
ISSN: 0969-8043
DOI: 10.1016/s0969-8043(97)00224-8

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## Abstract 4‐Fluoro‐__N__‐{2‐[4‐(6‐trifluoromethylpyridin‐2‐yl)piperazin‐1‐yl]ethyl}benzamide is a full 5‐HT~1A~ agonist with high affinity (__pK__~__i__~=9.3), selectivity and a __c__ log __P__ of 3.045. The corresponding PET radioligand 4‐[^18^F]fluoro‐__N__‐{2‐[4‐(6‐trifluoromethylpyridin‐2‐yl)