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[3H]UR-MK136: A Highly Potent and Selective Radioligand for Neuropeptide Y Y1 Receptors

✍ Scribed by Dr. Max Keller; Prof. Dr. Günther Bernhardt; Prof. Dr. Armin Buschauer

Book ID
102805524
Publisher
John Wiley and Sons
Year
2011
Tongue
English
Weight
667 KB
Volume
6
Category
Article
ISSN
1860-7179

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✦ Synopsis

Recently, we reported the bioisosteric substitution of a guanidine by an acylguanidine entity in argininamide-type neuropeptide Y (NPY) Y 1 receptor (Y 1 R) antagonists, such as BIBP 3226 [1] (1; Scheme 1), to be an effective strategy for the [a] Dr.

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