✦ LIBER ✦

[3H]U-69593 a highly selective ligand for the opioid κ receptor

✍ Scribed by Robert A. Lahti; Mary M. Mickelson; John M. McCall; Philip F. Von Voigtlander

Book ID: 115879338
Publisher: Elsevier Science
Year: 1985
Tongue: English
Weight: 255 KB
Volume: 109
Category: Article
ISSN: 0014-2999
DOI: 10.1016/0014-2999(85)90431-5

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

[3H]U-69593; a highly selective ligand f

[3H]U-69593; a highly selective ligand for the opioid κ receptor: R.A. Lahti, M.M. Mickelson, J.M. McCall and P.F. Vonvoigtlander, European J. Pharmacol. 109 (1985) 281–284

📂 Article 📅 1985 🏛 Elsevier Science 🌐 English ⚖ 35 KB

Ontogenesis of κ-opioid receptors in rat

Ontogenesis of κ-opioid receptors in rat brain using [3H]U-69593 as a binding ligand

✍ Ian Kitchen; Mary Kelly; M.Paz Viveros 📂 Article 📅 1990 🏛 Elsevier Science 🌐 English ⚖ 230 KB

Autoradiography of [3H]U-69593 binding s

Autoradiography of [3H]U-69593 binding sites in rat brain: evidence for κ opioid receptor subtypes

✍ Bruce Nock; Atul Rajpara; Lynn H. O'Connor; Theodore J. Cicero 📂 Article 📅 1988 🏛 Elsevier Science 🌐 English ⚖ 898 KB

ICI 197067 is a selective ligand for the

ICI 197067 is a selective ligand for the U-69593-sensitive κ opiate binding site

✍ Bruce Nock; Anthony L. Giordano; Theodore J. Cicero 📂 Article 📅 1989 🏛 Elsevier Science 🌐 English ⚖ 106 KB

A Kinetic Analysis of k-Opioid Agonist B

A Kinetic Analysis of k-Opioid Agonist Binding Using the Selective Radioligand [3H]U69593

✍ J. A. M. Smith; J. C. Hunter; R. G. Hill; J. Hughes 📂 Article 📅 1989 🏛 John Wiley and Sons 🌐 English ⚖ 994 KB

Synthesis of [3H]DIPPA: A potent irrever

Synthesis of [3H]DIPPA: A potent irreversible antagonist selective for the κ opioid receptor

✍ An-Chih Chang; Joseph D. Trometer; Philip S. Portoghese 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 French ⚖ 222 KB

## Abstract 2‐(3,4‐Dichlorophenyl)‐N‐methyl‐N‐[(1S)‐1‐(3‐isothiocyanatophenyl)‐2‐(1‐pyrrolidinyl)ethyl]acetamide (1, DIPPA) has been previously reported to be an opioid receptor affinity label that produces selective and long‐lasting κ opioid receptor antagonism in mice, High specific activity [^3^