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3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6

✍ Scribed by Mark E. Fraley; Justin T. Steen; Edward J. Brnardic; Kenneth L. Arrington; Keith L. Spencer; Barbara A. Hanney; Yuntae Kim; George D. Hartman; Steven M. Stirdivant; Bob A. Drakas; Keith Rickert; Eileen S. Walsh; Kelly Hamilton; Carolyn A. Buser; James Hardwick; Weikang Tao; Stephen C. Beck; Xianzhi Mao; Robert B. Lobell; Laura Sepp-Lorenzino; Youwei Yan; Mari Ikuta; Sanjeev K. Munshi; Lawrence C. Kuo; Constantine Kreatsoulas

Book ID: 108074154
Publisher: Elsevier Science
Year: 2006
Tongue: English
Weight: 248 KB
Volume: 16
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2006.08.118

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