✦ LIBER ✦

1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: Synthesis, pharmacological evaluation and mechanistic studies

✍ Scribed by Di Pietro, Ornella; Viayna, Elisabet; Vicente-García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, M. Victòria; Pérez, Belén; Andrisano, Vincenza; Luque, F. Javier; Lavilla, Rodolfo; Muñoz-Torrero, Diego

Book ID: 121448357
Publisher: Elsevier Science
Year: 2014
Tongue: French
Weight: 851 KB
Volume: 73
Category: Article
ISSN: 0223-5234
DOI: 10.1016/j.ejmech.2013.12.008

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

CoMFA, Synthesis, and Pharmacological Ev

CoMFA, Synthesis, and Pharmacological Evaluation of ( E )-3-(2-Carboxy-2-arylvinyl)-4,6-dichloro-1 H -indole-2-carboxylic Acids: 3-[2-(3-Aminophenyl)-2-carboxyvinyl]-4,6-dichloro-1 H -indole-2-carboxylic Acid, a Potent Selective Glycine-Site NMDA Receptor Antagonist †

✍ Baron, Bruce M.; Cregge, Robert J.; Farr, Robert A.; Friedrich, Dirk; Gross, Ray 📂 Article 📅 2005 🏛 American Chemical Society 🌐 English ⚖ 469 KB

ChemInform Abstract: Synthesis and in vi

ChemInform Abstract: Synthesis and in vitro and in vivo Evaluation of the 2-(6′Methoxy-3′,4′-dihydro-1′-naphthyl)-4H-3,1-benzoxazin-4-one as a New Potent Substrate Inhibitor of Human Leukocyte Elastase.

✍ Antonio Arcadi; Cinzia Asti; Laura Brandolini; Gianfranco Caselli; Fabio Marinel 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 29 KB 👁 2 views

Identification, Synthesis, and Biologica

Identification, Synthesis, and Biological Evaluation of 6-[(6 R )-2-(4-Fluorophenyl)-6-(hydroxymethyl)-4,5,6,7-tetrahydropyrazolo[1,5- a ]pyrimidin-3-yl]-2-(2-methylphenyl)pyridazin-3(2 H )-one (AS1940477), a Potent p38 MAP Kinase Inhibitor

✍ Asano, Toru; Yamazaki, Hitoshi; Kasahara, Chiyoshi; Kubota, Hirokazu; Kontani, T 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 906 KB

A New Series of N -[2,4-Dioxo-6- d -ribi

A New Series of N -[2,4-Dioxo-6- d -ribitylamino-1,2,3,4-tetrahydropyrimidin-5-yl]oxalamic Acid Derivatives as Inhibitors of Lumazine Synthase and Riboflavin Synthase: Design, Synthesis, Biochemical Evaluation, Crystallography, and Mechanistic Implications

✍ Zhang, Yanlei; Illarionov, Boris; Morgunova, Ekaterina; Jin, Guangyi; Bacher, Ad 📂 Article 📅 2008 🏛 American Chemical Society 🌐 English ⚖ 510 KB

Correction to Structure–Activity Relatio

Correction to Structure–Activity Relationship Study of N 6 -(2-(4-(1 H -Indol-5-yl)piperazin-1-yl)ethyl)- N 6 -propyl-4,5,6,7-tetrahydrobenzo[ d ]thiazole-2,6-diamine Analogues: Development of Highly Selective D3 Dopamine Receptor Agonists along with a Highly Potent D2/D3 Agonist and Their Pharmacological Characterization

✍ Johnson, Mark; Antonio, Tamara; Reith, Maarten E. A.; Dutta, Aloke K. 📂 Article 📅 2013 🏛 American Chemical Society 🌐 English ⚖ 197 KB

3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hyd

3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-alkylamides as a New Class of Synthetic Histone Deacetylase Inhibitors. 1. Design, Synthesis, Biological Evaluation, and Binding Mode Studies Performed through Three Different Docking Procedures

✍ Mai, Antonello; Massa, Silvio; Ragno, Rino; Cerbara, Ilaria; Jesacher, Florian; 📂 Article 📅 2003 🏛 American Chemical Society 🌐 English ⚖ 436 KB